Материал: MasterPass _ Pharmacology in 7 Days for Medical Students

CLASSIFICATIONS

•Enalapril

•Lisinopril

•Perindopril

•Quinapril

2Angiotensin II receptor blockers (competitive antagonists)

•Candesartan

•Eprosartan

•Irbesartan

•Losartan

•Sarasalin

•Telmisartan

•Valsartan

DSympathoplegics

1α and β blockers

•Carvedilol

•Labetalol

2α-adrenergic receptor antagonists

•Doxazosin

•Phentolamine

•Phenoxybenzmine

•Prazosin

•Terazosin

3Adrenergic neuron blockers

•Guanethidine

•Reserpine

4β-adrenergic receptor antagonists

•Atenolol

•Metoprolol

•Propranolol

5Centrally acting drugs

•Clonidine

•Guanabenz

•Guanfacine

•Methyldopa

6Ganglion-blocking drugs

•Trimethaphan

EVasodilators

1Arterial and venous

•Sodium nitroprusside

2Arterial

iOral

•Hydralazine

•Minoxidil

iiParenteral

•Diazoxide

•Fenoldopam

3Venodilators

•Nitroglycerin

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

Anti-Parkinsonian drugs

1 Dopaminergic drugs

aDopamine precursors

•Levodopa

bDopadecarboxylase inhibitors

•Carbidopa

•Benserazide

cDopamine releasing drugs

•Amantadine

2Dopaminergic agonist drugs a Ergot derivatives

•Bromocriptine

•Pergolide

bNon-ergot derivatives

•Pramipexole

•Ropinirole

3MAO-B inhibitors

•Selegiline

•Rasagiline

4Selective COMT (catechol-O-methyl transferase) inhibitors

•Tolcapone

•Entacapone

5Centrally acting antimuscarinics

•Biperidine

•Benzotropine

•Benzhexol

•Procyclidine

•Orphenadrine

6Other new approaches

aGene therapy

bSurgery

•Implantation of dopamine rich fragments of tissues, e.g. brain, adrenal glands.

•Thalomotomy

•Pallidotomy

•Thalamic stimulation by implanted electrodes

cFree radical scavengers

•Vitamin ‘E’

Antipeptic ulcer drugs

1 Antacids

aSystemic

•Sodium bicarbonate

bNon-systemic

iChemically acting

•Bismuth subcarbonate

•Calcium carbonate

•Magnesium carbonate

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CLASSIFICATIONS

•Magnesium hydroxide

•Magnesium oxide

iiPhysically acting

•Anion exchange resins

•Milk and mucin

iiiPhysico-chemically acting

•Aluminium hydroxide

•Aluminium phosphate

•Magnesium trisilicate

2 Anticholinergics

aNatural alkaloids

•Atropine

•Hyoscine

bSemi-synthetic

•Hyoscine butylbromide

cSelective anticholinergic

•Pirenzepine

dSynthetic

iQuartenary ammonium compounds

•Pipenzolate

•Propantheline

iiTertiary amines

•Dicyclomine

•Piperidolate

3Drugs for eradication of Helicobacter pylori

•Omeprazole and amoxycillin

•Omeprazole and clarithromycin

•Omeprazole, metronidazole, and clarithromycin/amoxycillin

•Bismuth sub-citrate, etronidazole and tetracycline/amoxycillin

4H2 receptor antagonists

•Cimetidine

•Famotidine

•Nizatidine

•Ranitidine

5Mucosal protective agents

aColloid bismuth compounds

•Bismuth subcitrate

bLiquorice derivatives

•Carbenoxolone

cProstaglandin analogue

•Misoprostol

dSulphated sucrose complex

•Sucralfate

6Proton pump inhibitors (PPIs)

•Esomeprazole

•Lansoprazole

•Omeprazole

•Pantoprazole

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

7Miscellaneous

•Metoclopramide

•Oxethezaine

•Proglumide

•Simethicone

Antipsychotic drugs

ATypical/classical antipsychotics

1Phenothiazine derivatives a Aliphatic compounds

•Promazine

•Chlorpromazine

bPiperazine compounds

•Perphenazine

•Fluphenazine

cPiperidine compounds

•Thioridazine

•Mesoridazine

2Butyrophenone derivatives

•Droperidol

•Haloperidol

3Thioxanthene derivatives

•Thiothixene

•Flupenthixol

4Rauwolfia alkaloids

•Reserpine

BAtypical/newer antipsychotics

•Aripiprazole

•Clozapine

•Olanzapine

•Quetiapine

•Loxapine

•Risperidone

•Ziprasidone

CDrugs used to treat manic-depressive disorders

•Carbamazepine

•Valproic acid

•Lamotrigine

•Lithium carbonate

Antithyroid drugs

1Thioamides

•Propyl thiouracil

•Methyl thiouracil

•Carbimazole

•Methimazole

2Anion inhibitors

•Potassium perchlorate

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CLASSIFICATIONS

•Thiocyanate

3 Iodides

•Lugol’s iodine

•Potassium iodide

4 Radio-active iodine

•I131

5β-adrenoceptor blockers

•Nadolol

•Propranolol

Beta-blocking drugs

AAccording to duration of action

1Intermediate acting

•Domolol

•Metoprolol

•Pindolol

•Propranolol

2Long acting

•Atenolol

•Bisoprolol

•Nadolol

3Ultrashort acting

•Esmolol

BAccording to β receptor selectivity

1Both α and β blockers

•Carvedilol

•Labetalol

2β1 blocker with partial β2 agonist activity

•Celiprolol

3β2 selective blocker

•Butoxamine

4Cardioselective (β1) blockers

iPure blockers

•Atenolol

•Bisoprolol

iiWith intrinsic sympathetic activity (ISA)

•Practalol

iiiWith membrane stabilising activity (MSA)

•Betaxolol

•Metoprolol

•Tolamolol

ivWith both ISA and MSA

•Acebutolol

5Non-selective (β1 and β2) blockers

iPure blockers

•Nadolol

•Sotalol

•Timolol

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