Материал: MasterPass _ Pharmacology in 7 Days for Medical Students

Внимание! Если размещение файла нарушает Ваши авторские права, то обязательно сообщите нам

PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

eOthers

Bupropion

Trazodone

5 Miscellaneous

• Alprazolam

• Flupenthixol

Antidiarrhoeal drugs

1Antimotility agents (drugs that prolong intestinal transit time by reducing motility)

a Anticholinergics

Atropine

Dicyclomine HCl

Propantheline

bBismuth subsalicylate

cNaturally occurring opium alkaloids

Codeine phosphate

dSynthetic opioid compounds

Diphenoxylate

Loperamide

2Adsorbants

Chalk

Charcoal

Isphagol husk

Kaolin

Methyl cellulose

Pectin

3Miscellaneous

Peppermint oil

Vegetable astringent

Anti-emetics

1Anticholinergics

Hyoscine

2Antihistamines (H1-antagonists)

Cyclizine

Hydroxyzine

Meclizine

Promethazine

Dimenhydrinate

Diphenhydramine

3Benzodiazepines

Diazepam

4Cannabinoids

Dronabinol

Nabilone

5D2-receptor antagonists

Domperidone

24

CLASSIFICATIONS

Metoclopramide

6 Glucocorticoids

Dexamethasone

Methylprednisolone

7Neurokinin-I-receptor-antagonists

Aprepitant

8Phenothiazines

Chlorpromazine

Prochlorperazine

Thiethylperazine

9Selective 5-HT3 receptor antagonists

Dolasetron

Granisetron

Ondansetron

Palonosetron

Antifungal drugs

1Drugs that disrupt fungal cell membrane A Polyenes

Amphotericin

Nystatin

BAzoles

iImidazoles

Ketoconazole

iiTriazoles

Fluconazole

iiiAllylamines

Terbinafine

2Drug that inhibits mitosis

Griseofulvin

3Drug that inhibits DNA synthesis

Flucytosine

Antimalarial drugs

AChemical classification

1Cinchona alkaloids

Quinine

2Diaminopyrimidine

Pyrimethamine

3Folate antagonists

Proguanil

44-Aminoquinolines

Amodiaquine

Chloroquine

58-Aminoquinolines

Primaquine

6Quinoline methanol

Mefloquine

25

PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

• Quinidine

7Sulfonamides

Sulphadoxine

8Sulphones

Dapsone

9Tetracyclines

Doxycycline

10Miscellaneous

Halofantrin

Qinghaosu derivatives (artemisinins), i.e. artemether and artisunate

11Combinations

Fansidar (pyrimethamine + sulfadoxine)

Fansimef (pyrimethamine + sulfadoxine + mefloquine)

Maloprim (pyrimethamine + dapsone)

Malarone (atovaquone + proguanil)

BClassification based on site of action

1Tissue schizonticides (acting on hepatic cycle: pre-erythrocytic stage) a Against primary tissue forms for causal prophylaxis

• Proguanil

bAgainst latent tissue forms, for terminal prophylaxis/radical cure

Primaquine

2Blood schizonticides (acting on erythrocytic cycle for suppressive cure) a Rapidly acting blood schizonticides

Artemisinins

Amodiaquine

Chloroquine

Halofantrin

Mefloquine

Quinine

bSlower acting blood schizonticides

Doxycycline

Proguanil

Pyrimethamine

3Gametocides against sexual erythrocytic forms

Primaquine (against plasmodium falciparum)

Chloroquine and quinine (against plasmodium vivax and ovale)

Antigout drugs

ADrugs for acute attack

1Natural alkaloids

Colchicine

Demecolchicine

2NSAIDs specially used in gout

Fenoprofen

Indomethacine

Naproxen

Oxaprozin

Oxyphenbutazone

26

CLASSIFICATIONS

Phenylbutazone

Piroxicam

3Corticosteroids

Hydrocortisone

Prednisolone

BDrugs for chronic gout

1Drugs which increase excretion of uric acid (uricosuric agents)

Aspirin (in high doses)

Oxyphenbutazone

Phenylbutazone

Probenecid

Sulfinpyrazone

2Drugs which decrease synthesis of uric acid (xanthine oxidase inhibitors)

Allopurinol

Antihelminthic drugs

1Drugs acting against nematodes

Albendazole

Mebendazole

Thiabendazole

Diethyl carbamazine

Pyrantel pamoate

2Drugs acting against trematodes

Praziquantel

3Drugs acting against cestodes

Niclosamide

Drugs used in the Rx of leprosy

Clofazimine

Dapsone

Fluoroquinolones

Macrolides

Minocycline

Rifampicin

Miscellaneous:

Ethionamide

Thalidomide

Drugs used in the Rx of tuberculosis

1First-line drugs

Ethambutol

Isoniazid

Pyrazinamide

Rifampin

Streptomycin

2Second-line drugs

Alikacin and kanamycin

27

PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

Ciprofloxacin, levofloxacin and ofloxacin

Capreomycin

Cycloserine

Ethionamide

Rifabutin

Rifapentine

Antihypertensive drugs

ACalcium channel blockers

1Benzothiazepines

Diltiazem

2Diarylaminopropylamine

Bepridil

3Dihydropyridines

Amlodipine

Felodipine

Isradipine

Nicardipine

Nifedipine

Nimodipine

Nisoldipine

Nitrendipine

4Diphenylpiperazines

Flunarizine

Ranolazine

Trimetazidine

5Phenyl Alkylamines

Gallopamil

Verapamil

BDiuretics

1Loop diuretics

Bumetanide

Ethacrynic acid

Furosemide

2Potassium-sparing diuretics

Amiloride

Spironolactone

Triamterene

3Thiazides and related agents

Benzthiazide

Chlorthalidone

Chlorothiazide

Hydrochlorothiazide

Indapamide

CDrugs acting on renin-angiotensin system

1Angiotensin converting enzyme (ACE) inhibitors

Benzapril

Captopril

28