Материал: MasterPass _ Pharmacology in 7 Days for Medical Students

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

Newer drugs:

1GABA analogue

Gabapentin

Vigabatrin

2Miscellaneous

Lamotrigine

Felbamate

Topiramate

Older drugs:

1Bromides

Sodium and Potassium bromide

2Carbonic anhydrase inhibitors

Acetazolamide

3Oxazolidinedione derivatives

Trimethadione

4Miscellaneous

Paraldehyde

Adrenocorticosteroids

Natural

1Glucocorticoids

Cortisol

Corticosterone

2Mineralocorticoids

Aldosterone

11-Deoxy corticosterone acetate

Synthetic

1Glucocorticoids

Cortisone

Prednisone

Prednisolone

Methylprednisolone

Paramethasone

Dexamethasone

Triamcinolone

Betamethasone valerate

Beclomethasone dipropionate

2Mineralocorticoids

1 Fludrocortisone

Antiviral drugs

1Agents to treat herpes simplex virus (HSV) and varicella-zoster virus (VSV) infections (DNA-polymerase inhibitors)

Acyclovir

Valacyclovir

Famciclovir

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CLASSIFICATIONS

Penciclovir

Foscarnet

Trifluridine

2Agents to treat cytomegalovirus (CMV) infections

Cidofovir

Foscarnet

Fomivirsen

Ganciclovir

Valganciclovir

3Antiretroviral agents

iNucleoside reverse transcriptase inhibitors (NRTIs)

Abacavir

Didanosine

Lamivudine

Stavudine

Zidovudine

Zalcitabine

iiNon-nucleoside reverse transcriptase inhibitors (NNRTIs)

Delavirdine

Efavirenz

Nevirapine

iiiProtease inhibitors

Amprenavir

Indinavir

Nelfinavir

Ritonavir

Saquinavir

ivFusion inhibitors

Enfuvirtide

4Antihepatitis agents

Adefovir

Interferon

Lamivudine

Ribavirin

5Anti-influenza agents

Amantadine

Rimantadine

Oseltamivir

Zanamivir

NSAIDs

ADrugs with analgesic and marked anti-inflammatory effects

1Salicylic acid derivatives

Aspirin (acetyl salicylic acid)

Salicylic acid

Sodium salicylate

Methyl salicylate

Choline salicylate

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

Magnesium salicylate

Diflunisal

Benorylate

2Pyrazolone derivatives

Phenylbutazone

Oxyphenbutazone

Azapropazone

3Acetic acid derivatives

Diclofenac

Indomethacin

Tolmetin

Sulnidac

Etodolac

4Oxicams

Piroxicam

Meloxicam

5Miscellaneous

Nimuselide

Celecoxib

Rofecoxib

BDrugs with analgesic and moderate anti-inflammatory effects

1Propionic acid derivatives

Ibuprofen

Ketoprofen

Fenoprofen

Flurbiprofen

Carprofen

Indoprofen

Naproxen

Oxaprozin

2Fenamic acid derivatives

Mefenamic acid

Meclofenamic acid

Flufenamic acid

Tolfenamic acid

CDrugs with analgesic and weak anti-inflammatory effects

Paracetamol (aniline derivative)

Adrenergic neuron blockers

1Drugs which interfere with synthesis of noradrenaline

Metyrosine (alpha-methyl tyrosine)

2Drugs that inhibit storage of noradrenaline

Deserpidine

Reserpine

3Drugs that prevent release of noradrenaline

Bethanidine

Debrisoquin

Guanadrel

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CLASSIFICATIONS

Guanethidine

Guanoxan

Alpha-adrenergic blockers

AChemical classification

1Beta-haloalkylamines

Dibenamine

Phenoxybenzamine

2Benzodioxans

Dibuzaine

Diperoxan

3Benzene sulfonamide

Tamsulosin

4Dibenzapines

Azepetine

5Ergot alkaloid

Dihydroergotamine

Ergotamine

6Phenothiazines

Chlorpromazine

7Phenoxyalkylamines

Thymoxamine

8Piperazinyl quinazolines

Doxazosin

Prazosin

Terazosin

9Substituted imidazolines

Phentolamine

Tolazoline

10Miscellaneous

Carvedilol

Indoramin

Labetalol

BAccording to reversibility of action

1Irreversible (non-competitive blockers; long-acting)

Dibenamine

Phenoxybenzamine

2Reversible (competitive blockers; short-acting)

Doxazosin

Prazosin

Phentolamine

Terazosin

Tolazoline

Trimazosin

Urapidil

CAccording to receptor selectivity

1Mixed α and β adrenoceptor blocking drugs

Carvedilol

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

• Labetalol

2Selective α-blockers

iα1-blockers

Alfuzosin

Doxazosin

Pinacidal

Prazosin

Tamsulosin

Teruzosin

Trimazosin

iiα2-blockers

Idazoxan

Yohimbine

3Non-selective (both α1 and α2-blockers)

Dibenamine

Dihydroergotamine

Ergotamine

Phentolamine

Phenoxybenzamine

Tolazoline

Aminoglycosides

1Natural

Gentamycin

Kanamycin

Neomycin

Streptomycin

Tobramycin

2Semi-synthetic

Amikacin

Netilmicin

Members of macrolide group

Azithromycin

Clarithromycin

Roxithromycin

Telithromycin

Carbomycin

Erythromycin

Oleandomycin

Spiramycin

Amoebicides

AChemical classification

1Dichloroacetamides

Clefamide

Etofamide

Diloxanide furoate

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