PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS
Newer drugs:
1GABA analogue
•Gabapentin
•Vigabatrin
2Miscellaneous
•Lamotrigine
•Felbamate
•Topiramate
Older drugs:
1Bromides
•Sodium and Potassium bromide
2Carbonic anhydrase inhibitors
•Acetazolamide
3Oxazolidinedione derivatives
•Trimethadione
4Miscellaneous
•Paraldehyde
Adrenocorticosteroids
Natural
1Glucocorticoids
•Cortisol
•Corticosterone
2Mineralocorticoids
•Aldosterone
•11-Deoxy corticosterone acetate
Synthetic
1Glucocorticoids
•Cortisone
•Prednisone
•Prednisolone
•Methylprednisolone
•Paramethasone
•Dexamethasone
•Triamcinolone
•Betamethasone valerate
•Beclomethasone dipropionate
2Mineralocorticoids
1 Fludrocortisone
Antiviral drugs
1Agents to treat herpes simplex virus (HSV) and varicella-zoster virus (VSV) infections (DNA-polymerase inhibitors)
•Acyclovir
•Valacyclovir
•Famciclovir
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CLASSIFICATIONS
•Penciclovir
•Foscarnet
•Trifluridine
2Agents to treat cytomegalovirus (CMV) infections
•Cidofovir
•Foscarnet
•Fomivirsen
•Ganciclovir
•Valganciclovir
3Antiretroviral agents
iNucleoside reverse transcriptase inhibitors (NRTIs)
•Abacavir
•Didanosine
•Lamivudine
•Stavudine
•Zidovudine
•Zalcitabine
iiNon-nucleoside reverse transcriptase inhibitors (NNRTIs)
•Delavirdine
•Efavirenz
•Nevirapine
iiiProtease inhibitors
•Amprenavir
•Indinavir
•Nelfinavir
•Ritonavir
•Saquinavir
ivFusion inhibitors
•Enfuvirtide
4Antihepatitis agents
•Adefovir
•Interferon
•Lamivudine
•Ribavirin
5Anti-influenza agents
•Amantadine
•Rimantadine
•Oseltamivir
•Zanamivir
NSAIDs
ADrugs with analgesic and marked anti-inflammatory effects
1Salicylic acid derivatives
•Aspirin (acetyl salicylic acid)
•Salicylic acid
•Sodium salicylate
•Methyl salicylate
•Choline salicylate
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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS
•Magnesium salicylate
•Diflunisal
•Benorylate
2Pyrazolone derivatives
•Phenylbutazone
•Oxyphenbutazone
•Azapropazone
3Acetic acid derivatives
•Diclofenac
•Indomethacin
•Tolmetin
•Sulnidac
•Etodolac
4Oxicams
•Piroxicam
•Meloxicam
5Miscellaneous
•Nimuselide
•Celecoxib
•Rofecoxib
BDrugs with analgesic and moderate anti-inflammatory effects
1Propionic acid derivatives
•Ibuprofen
•Ketoprofen
•Fenoprofen
•Flurbiprofen
•Carprofen
•Indoprofen
•Naproxen
•Oxaprozin
2Fenamic acid derivatives
•Mefenamic acid
•Meclofenamic acid
•Flufenamic acid
•Tolfenamic acid
CDrugs with analgesic and weak anti-inflammatory effects
•Paracetamol (aniline derivative)
Adrenergic neuron blockers
1Drugs which interfere with synthesis of noradrenaline
•Metyrosine (alpha-methyl tyrosine)
2Drugs that inhibit storage of noradrenaline
•Deserpidine
•Reserpine
3Drugs that prevent release of noradrenaline
•Bethanidine
•Debrisoquin
•Guanadrel
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CLASSIFICATIONS
•Guanethidine
•Guanoxan
Alpha-adrenergic blockers
AChemical classification
1Beta-haloalkylamines
•Dibenamine
•Phenoxybenzamine
2Benzodioxans
•Dibuzaine
•Diperoxan
3Benzene sulfonamide
•Tamsulosin
4Dibenzapines
•Azepetine
5Ergot alkaloid
•Dihydroergotamine
•Ergotamine
6Phenothiazines
•Chlorpromazine
7Phenoxyalkylamines
•Thymoxamine
8Piperazinyl quinazolines
•Doxazosin
•Prazosin
•Terazosin
9Substituted imidazolines
•Phentolamine
•Tolazoline
10Miscellaneous
•Carvedilol
•Indoramin
•Labetalol
BAccording to reversibility of action
1Irreversible (non-competitive blockers; long-acting)
•Dibenamine
•Phenoxybenzamine
2Reversible (competitive blockers; short-acting)
•Doxazosin
•Prazosin
•Phentolamine
•Terazosin
•Tolazoline
•Trimazosin
•Urapidil
CAccording to receptor selectivity
1Mixed α and β adrenoceptor blocking drugs
•Carvedilol
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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS
• Labetalol
2Selective α-blockers
iα1-blockers
•Alfuzosin
•Doxazosin
•Pinacidal
•Prazosin
•Tamsulosin
•Teruzosin
•Trimazosin
iiα2-blockers
•Idazoxan
•Yohimbine
3Non-selective (both α1 and α2-blockers)
•Dibenamine
•Dihydroergotamine
•Ergotamine
•Phentolamine
•Phenoxybenzamine
•Tolazoline
Aminoglycosides
1Natural
•Gentamycin
•Kanamycin
•Neomycin
•Streptomycin
•Tobramycin
2Semi-synthetic
•Amikacin
•Netilmicin
Members of macrolide group
•Azithromycin
•Clarithromycin
•Roxithromycin
•Telithromycin
•Carbomycin
•Erythromycin
•Oleandomycin
•Spiramycin
Amoebicides
AChemical classification
1Dichloroacetamides
•Clefamide
•Etofamide
•Diloxanide furoate
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